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Publikace

Published in Top 10% journals in the field

MISTRÍK, M., Z. ŠKROTT, P. MULLER, A. PANACEK, L. HOCHVALDOVA, K. CHROMÁ, T. BUCHTOVÁ, V. VANDOVA, L. KVÍTEK, J. BÁRTEK
Microthermal-induced subcellular-targeted protein damage in cells on plasmonic nanosilver-modified surfaces evokes a two-phase HSP-p97/VCP response. Nature Communications. 2021, 12(1), 713, ISSN: 2041-1723, PMID: 33514738,
GONZALES, G., J. HODOŇ, A. KAZAKOVA, C. D´ACUNTO, P. KANOVSKY, M. URBAN, M. STRNAD
Novel pentacyclic triterpenes exhibiting strong neuroprotective activity in SH-SY5Y cells in salsolinol- and glutamate-induced neurodegeneration models. European Journal of Medicinal Chemistry. 2021, 213, 113168, ISSN: 0223-5234, PMID: 33508480,
VANDA, D., V. CANALE, S. CHAUMONT-DUBEL, R. KURCZAB, G. SATALA, K. P., M. KRAWCZYK, W. PIETRUS, K. BLICHARZ, E. PEKALA, A. BOJARSKI, P. POPIK, P. MARIN, M. SOURAL, P. ZAJDEL
Imidazopyridine-Based 5-HT 6 Receptor Neutral Antagonists: Impact of N1-Benzyl and N1-Phenylsulfonyl Fragments on Different Receptor Conformational States. Journal of Medicinal Chemistry. 2021, 64(2), 1180-1196, ISSN: 0022-2623, PMID: 33439019,
CReM: chemically reasonable mutations framework for structure generation. Journal of Cheminformatics. 2020, 12(1), 28, ISSN: 1758-2946, PMID: 33430959,
URBAN, M., V. ŠLACHTOVÁ, L. BRULÍKOVÁ
Small organic molecules targeting the energy metabolism of Mycobacterium tuberculosis. European Journal of Medicinal Chemistry. 2021, 212, 113139, ISSN: 0223-5234, PMID: 33422979,
KRAJČOVIČOVÁ, S., R. JORDA, D. VANDA, M. SOURAL, V. KRYŠTOF
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton's tyrosine kinase. European Journal of Medicinal Chemistry. 2020, 211, 113094, ISSN: 0223-5234, PMID: 33340912,
SVEC, P., Z. NOVÝ, J. KUCKA, M. PETŘÍK, O. SEDLACEK, M. KUCHAR, B. LIŠKOVÁ, M. MEDVEDÍKOVÁ, K. KOLOUCHOVA, O. GROBORZ, L. LOUKOTOVA, R. KONEFAL, M. HAJDÚCH, M. HRUBY
Iodinated Choline Transport-Targeted Tracers. Journal of Medicinal Chemistry. 2020, 63(24), 15960–15978, ISSN: 0022-2623, PMID: 33271015,
CHASÁK, J., V. ŠLACHTOVÁ, M. URBAN, L. BRULÍKOVÁ
Squaric acid analogues in medicinal chemistry. European Journal of Medicinal Chemistry. 2021, 209, 112872, ISSN: 0223-5234, PMID: 33035923,
RUČILOVÁ, V., A. SWIERRCZEK, D. VANDA, P. FUNK, B. LEMROVÁ, A. GAWALSKA, A. BUCKI, B. NOWAK, M. ZADROZNA, K. POCIECHA, M. SOURAL, E. WYSKA, M. PAWLOWSKI, G. CHLON-RZEPA, P. ZAJDEL
New imidazopyridines with phosphodiesterase 4 and 7 inhibitory activity and their efficacy in animal models of inflammatory and autoimmune diseases. European Journal of Medicinal Chemistry. 2020, 209, 112854, ISSN: 0223-5234, PMID: 33022582,
SVOBODOVÁ, L., M. DVORAKOVA, M. RUCKI, K. KEJLOVA, H. KANDAROVA, H. KOLÁŘOVÁ, M. MANNERSTROM, T. HEINONEN
Safety testing of adult novelties using in vitro methods. Regulatory Toxicology and Pharmacology. 2020, 117, 104780, ISSN: 0273-2300, PMID: 32898621,