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Publikace

Published in Top 10% journals in the field

YANG, C., L. POSTOVA SLAVETINSKA, M. FLEUTI, B. KLEPETAROVA, M. TICHÝ, S. GURSKÁ, P. PAVLIŠ, P. DŽUBÁK, M. HAJDÚCH, M. HOCEK
Synthesis of Polycyclic Hetero-Fused 7-Deazapurine Heterocycles and Nucleosides through C-H Dibenzothiophenation and Negishi Coupling. Journal of the American Chemical Society. 2022, 144(42), 19437-19446, ISSN: 0002-7863, PMID: 36245092,
ŘEZNÍČKOVÁ, E., S. KRAJČOVIČOVÁ, M. PERINA, A. KOVALOVA, M. SOURAL, V. KRYŠTOF
Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC). European Journal of Medicinal Chemistry. 2022, 243, 114792, ISSN: 0223-5234, PMID: 36191408,  PDF.
HODOŇ, J., I. FRYDRYCH, Z. TRHLÍKOVÁ, J. POKORNÝ, L. BORKOVÁ, S. BENICKÁ, M. VLK, B. LIŠKOVÁ, A. KUBÍČKOVÁ, M. MEDVEDÍKOVÁ, M. PISÁR, J. ŠAREK, V. DAS, A. LIGASOVÁ, K. KOBERNA, P. DŽUBÁK, M. HAJDÚCH, M. URBAN
Triterpenoid pyrazines and pyridines - Synthesis, cytotoxicity, mechanism of action, preparation of prodrugs. European Journal of Medicinal Chemistry. 2022, 243, 114777, ISSN: 0223-5234, PMID: 36174412,  PDF.
JORDA, R., L. HAVLÍČEK, M. PERINA, V. VOJÁČKOVÁ, T. POSPÍŠIL, S. DJUKIC, J. SKERLOVA, J. GRÚZ, N. RENESOVA, P. KLENER, P. ŘEZÁČOVÁ, M. STRNAD, V. KRYŠTOF
3,5,7-Substituted Pyrazolo[4,3- d]Pyrimidine Inhibitors of Cyclin-Dependent Kinases and Cyclin K Degraders. Journal of Medicinal Chemistry. 2022, 65(13), 8881-8896, ISSN: 0022-2623, PMID: 35749742,
SIKOROVÁ, K., S. MOON, H. YOON, A. STRNAD, J. SONG, M. PETŘEK
HLA class II variants defined by next generation sequencing are associated with sarcoidosis in Korean patients. Scientific Reports. 2022, 12(1), 9302, ISSN: 2045-2322, PMID: 35661780,
KLOS, D., M. DUŠEK, E. SAMOLOVA, M. ZATLOUKAL, V. NOZKOVA, N. NESNAS, L. PLACKOVA, R. KOPRNA, Z. SPISEK, H. VYLICILOVA, O. PLIHAL, K. DOLEZAL, J. VOLLER, A. KADLECOVA, M. STRNAD, L. PLÍHALOVÁ
New Water-Soluble Cytokinin Derivatives and Their Beneficial Impact on Barley Yield and Photosynthesis. Journal of Agricultural and Food Chemistry. 2022, 70(23), 7288-7301, ISSN: 0021-8561, PMID: 35658447,
ZACHOVÁ, K., J. JEMELKOVA, P. KOSZTYU, Y. OHYAMA, K. TAKAHASHI, J. ZADRAZIL, J. ORSAG, K. MATOUSOVIC, D. GALUSZKOVÁ, N. PETEJOVA, J. MESTECKY, M. RAŠKA
Galactose-Deficient IgA1 B cells in the Circulation of IgA Nephropathy Patients Carry Preferentially Lambda Light Chains and Mucosal Homing Receptors. Journal of the American Society of Nephrology. 2022, 33(5), 908-917, ISSN: 1046-6673, PMID: 35115327,
WOLRAB, D., R. JIRASKO, E. CIFKOVA, M. HORING, D. MEI, M. CHOCHOLOUSKOVA, O. PETERKA, J. IDOWIAK, T. HRNCIAROVA, L. KUCHAR, R. AHRENDS, R. BRUMAROVÁ, D. FRIEDECKÝ, G. VIVO-TRUYOLS, P. SKRHA, J. SKRHA, R. KUCERA, B. MELICHAR, G. LIEBISCH, R. BURKHARDT, M. WENK, A. CAZENAVE-GASSIOT, P. KARASEK, I. NOVOTNY, K. GREPLOVA, R. HRSTKA, M. HOLCAPEK
Lipidomic profiling of human serum enables detection of pancreatic cancer. Nature Communications. 2022, 13(1), 124, ISSN: 2041-1723, PMID: 35013261,
RAFFAELE, M., K. KOVACOVICOVA, T. BIAGINI, O. LO RE, J. FROHLICH, S. GIALLONGO, J. NHAN, A. GIANNONE, D. CABIBI, M. IVANOV, A. TONCHEV, M. MISTRÍK, M. LACEY, P. DŽUBÁK, S. GURSKÁ, M. HAJDÚCH, J. BÁRTEK, T. MAZZA, V. MICALE, S. CURRAN, M. VINCIGUERRA
Nociceptin/orphanin FQ opioid receptor (NOP) selective ligand MCOPPB links anxiolytic and senolytic effects. Geroscience. 2021, 44(1), 463-483, ISSN: 2509-2715, PMID: 34820764,
MOUDRÝ, P., K. CHROMÁ, S. BURSAC, S. VOLAREVIC, J. BÁRTEK
RNA-interference screen for p53 regulators unveils a role of WDR75 in ribosome biogenesis. Cell Death and Differentiation. 2022, 29(3), 687-696, ISSN: 1350-9047, PMID: 34611297,