Publications

Published in Top 10% journals in the field

JORDA, R., S. KRAJČOVIČOVÁ, P. KRÁLOVÁ, M. SOURAL, V. KRYŠTOF
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome. European Journal of Medicinal Chemistry. 2020, 204, 112636, ISSN: 0223-5234, PMID: 32731189,
DVOŘANOVÁ ŠTĚPÁNKOVÁ, J., M. KUGLER, J. HOLUB, V. SICHA, V. DAS, J. NEKVINDA, S. EL ANWAR, M. HAVRANEK, K. POSPISILOVA, M. FABRY, V. KRAL, M. MEDVEDÍKOVÁ, S. MATEJKOVA, B. LIŠKOVÁ, S. GURSKÁ, P. DŽUBÁK, J. BRYNDA, M. HAJDÚCH, B. GRUNER, P. ŘEZÁČOVÁ
Sulfonamido Carboranes as Highly Selective Inhibitors of Cancer-Specific Carbonic Anhydrase IX. European Journal of Medicinal Chemistry. 2020, 200, 112460, ISSN: 0223-5234, PMID: 32505851,
KEJLOVA, K., H. BENDOVA, J. CHRZ, M. DVORAKOVA, L. SVOBODOVÁ, A. VLKOVA, L. KUBAC, R. KORINKOVA, J. CERNY, D. OCADLIKOVA, M. RUCKI, T. HEINONEN, D. JIROVA, S. LETASIOVA, H. KANDAROVA, H. KOLÁŘOVÁ
Toxicological Testing of a Photoactive Phthalocyanine-Based Antimicrobial Substance. Regulatory Toxicology and Pharmacology. 2020, 115, 104685, ISSN: 0273-2300, PMID: 32454236,
CHYRA, Z., T. SEVCIKOVA, P. VOJTA, J. PUTEROVA, L. BROZOVA, K. GROWKOVA, J. FILIPOVA, M. ZATOPKOVA, S. GROSICKI, A. BARCHNICKA, W. JEDRZEJCAK, A. WASCUK-GAJDA, A. JUNGOVA, A. MIKULASOVA, M. HAJDÚCH, M. MOKREJS, L. POUR, M. STORK, L. HARVANOVA, M. MISTRÍK, G. MIKALA, P. ROBAK, A. CZYZ, J. DEBSKI, L. USNARSKA-ZUBKIEWICZ, A. JURCZYSZYN, L. STEJSKAL, G. MORGAN, F. KRYUKOV, E. BUDINSKA, M. SIMICEK, T. JELINEK, M. HRDINKA, R. HAJEK
Heterogenous mutation spectrum and deregulated cellular pathways in aberrant plasma cells underline molecular pathology of light-chain amyloidosis. Haematologica. 2020, 106(2), 601-604, ISSN: 0390-6078, PMID: 32381580,
FIEDLER, J., M. REISER, P. KOSTAL, J. KUBALE, S. OSTRY, T. HRBAC, P. KESNEROVA, T. FADRNA, K. LANGOVÁ, R. HERZIG, D. SKOLOUDIK
Blood Flow Volume Measurement in Cervical and Intracranial Arteries using Quantitative Magnetic Resonance Angiography and Duplex Sonography (Bocaccia) - A Prospective Observational Study. Ultraschall in der Medizin. 2020, 42(1), 65-74, ISSN: 0172-4614, PMID: 32340045,
ŘEHULKA, J., K. BÜRGLOVÁ, P. KREJČÍ, S. GURSKÁ, P. HRADIL, M. HAJDÚCH, P. DŽUBÁK, J. HLAVÁČ
Fluorinated derivatives of 2-phenyl-3-hydroxy-4(1H)-quinolinone as tubulin polymerization inhibitors. European Journal of Medicinal Chemistry. 2020, 192, 112176, ISSN: 0223-5234, PMID: 32120327,
SAID, M., W. ELDEHNA, A. NOCENTINI, S. FAHIM, A. BONARDI, A. ELGAZAR, V. KRYŠTOF, D. SOLIMAN, H. ABDEL-AZIZ, P. GRATTERI, S. ABOU-SERI, C. SUPURAN
Sulfonamide-based ring-fused analogues for CAN508 as novel carbonic anhydrase inhibitors endowed with antitumor activity: Design, synthesis, and in vitro biological evaluation. European Journal of Medicinal Chemistry. 2020, 189(2020), 112019, ISSN: 0223-5234, PMID: 31972394,
JORDA, R., P. MAGAR, D. HENDRYCHOVA, K. PAUK, M. DIBUS, E. PILAROVA, A. IMRAMOVSKY, V. KRYŠTOF
Novel modified leucine and phenylalanine dipeptides modulate viability and attachment of cancer cells. European Journal of Medicinal Chemistry. 2020, 188, 112036, ISSN: 0223-5234, PMID: 31931341,
BORKOVÁ, L., I. FRYDRYCH, N. JAKUBCOVÁ, R. ADÁMEK, B. LIŠKOVÁ, S. GURSKÁ, M. MEDVEDÍKOVÁ, M. HAJDÚCH, M. URBAN
Synthesis and biological evaluation of triterpenoid thiazoles derived from betulonic acid, dihydrobetulonic acid, and ursonic acid. European Journal of Medicinal Chemistry. 2019, 185, 111806, ISSN: 0223-5234, PMID: 31677446,
GRUNER, B., J. BRYNDA, V. DAS, V. SICHA, J. ŠTĚPÁNKOVÁ, J. NEKVINDA, J. HOLUB, K. POSPISILOVA, M. FABRY, P. PACHL, V. KRAL, M. KUGLER, V. MAŠEK, M. MEDVEDÍKOVÁ, S. MATEJKOVA, A. NOVÁ, B. LIŠKOVÁ, S. GURSKÁ, P. DŽUBÁK, M. HAJDÚCH, P. ŘEZÁČOVÁ
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX. Journal of Medicinal Chemistry. 2019, 62(21), 9560-9575, ISSN: 0022-2623, PMID: 31568723,